SCHEMBL7069359

SCHEMBL7069359

Cc1nc(-c2ccc(C(=O)N3CCN(S(=O)(=O)c4ccc(Cl)c(Cl)c4)CC3)cc2)no1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.48
ATM Q13315 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
LMNA P02545 4/20 0.47
F10 P00742 2/20 0.47
MGLL Q99685 1/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
TP53 P04637 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8072947 0.96 THRB (0.46) THRBATMSMN1; SMN2CYP2D6CYP2C9
SCHEMBL7074664 0.94 THRB (0.53) THRBATMSMN1; SMN2CYP2D6CYP2C9
SCHEMBL7071746 0.90 MEN1 (0.54) SMN1; SMN2CYP2D6CYP2C9CYP2C19LMNA
SCHEMBL7070562 0.89 F10 (0.57) ATMF10
SCHEMBL7069907 0.89 VCAM1 (0.52) ATMSMN1; SMN2LMNAMGLLMEN1
SCHEMBL7071596 0.88 LMNA (0.54) THRBSMN1; SMN2CYP2D6CYP2C9CYP2C19
SCHEMBL7074109 0.88 ALDH1A1 (0.48) THRBSMN1; SMN2CYP2D6CYP2C9CYP2C19
SCHEMBL7074222 0.88 LMNA (0.62) THRBSMN1; SMN2CYP2D6CYP2C9CYP2C19
SCHEMBL7074230 0.87 HPGD (0.53) SMN1; SMN2LMNAMGLLALDH1A1
SCHEMBL7076713 0.87 RAB9A (0.54) THRBATMSMN1; SMN2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed