SCHEMBL8076141

SCHEMBL8076141

Cc1ccc(-c2sccc2C)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 8/20 0.55
CYP3A4 P08684 3/20 0.53
CYP2C19 P33261 3/20 0.53
CYP2B6 P20813 2/20 0.53
CYP2E1 P05181 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
PTGS2 P35354 1/20 0.49
PGR P06401 2/20 0.45
CASP3 P42574 1/20 0.41
NISCH Q9Y2I1 1/20 0.40
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
XBP1 P17861 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ACHE P22303 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13130594 0.93 CYP2A6 (0.61) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL14640117 0.82 CYP2A6 (0.52) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL2122531 0.82 CYP2A6 (0.58) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL28479595 0.82 CYP2A6 (0.52) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL10407505 0.82 CYP2A6 (0.52) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL693906 0.82 CYP2A6 (0.59) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL1821918 0.81 CYP2A6 (0.60) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL29018974 0.80 CYP2A6 (0.50) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1
SCHEMBL28228496 0.79 PTGS2 (0.71) PTGS2
SCHEMBL722595 0.79 CYP2A6 (0.56) CYP2A6CYP3A4CYP2C19CYP2B6CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10460879-B2 Photoelectric conversion element, dye-sensitized solar cell, metal complex dye, dye solution, dye-adsorbed electrode, and method for producing dye-sensitized solar cell FUJIFILM CORPORATION (JP) 2019-10-29 US disclosed
US-8063099-B2 Trans-3-aza-bicyclo[3.1.0]hexane derivatives ACTELION PHARMACEUTICALS LTD. (CH) 2011-11-22 US disclosed
US-8003626-B2 in particular fungicidally active; use in agriculture or horticulture for controlling/preventing infestation of plants by phytopathogens; 1-methyl-3-trifluoromethyl-4,5-dihydro-1H-pyrazole-4-carboxylic acid [2-(1,3-dimethyl-butyl)-thiophen-3-yl]-amide SYNGENTA CROP PROTECTION, INC. (US) 2011-08-23 US disclosed
EP-2185512-B1 TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-12-29 EP disclosed
US-20100204285-A1 TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD. (CH) 2010-08-12 US disclosed
WO-2009016560-A2 TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2009-02-05 WO disclosed
US-20080188442-A1 Pyrazole-4-Carboxamide Derivatives as Microbiocides SYNGENTA CROP PROTECTION, INC. (US) 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188442-A1 Pyrazole-4-Carboxamide Derivatives as Microbiocides CD14, FPR1, FPR2 CYP2A6 234/4885CYP3A4 38/4885CYP2C19 59/4885
US-20100204285-A1 TRANS-3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES HCRTR1, HCRTR2, CNR1 CYP2A6 512/4885CYP3A4 500/4885CYP2C19 447/4885
US-10460879-B2 Photoelectric conversion element, dye-sensitized solar cell, metal complex dye, dye solution, dye-adsorbed electrode, and method for producing dye-sensitized solar cell CHRM1, L1CAM, CRY1 CYP2A6 3345/4885CYP3A4 2894/4885CYP2C19 3657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.