SCHEMBL8076664

SCHEMBL8076664

CCOC(=O)[C@@H]1OS(=O)(=O)OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.37
POLB P06746 1/20 0.36
PPM1B O75688 1/20 0.33
PTPN1 P18031 1/20 0.33
PPP1CC P36873 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 4/20 0.32
GAA P10253 1/20 0.32
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8076662 1.00 LMNA (0.37) LMNAPOLBPPM1BPTPN1PPP1CC
SCHEMBL900783 0.77 LMNA (0.43) LMNAPOLBPPM1BPTPN1PPP1CC
SCHEMBL17577372 0.72 TSHR (0.46) LMNAPPM1BPTPN1PPP1CCTSHR
SCHEMBL18166910 0.72 TSHR (0.46) LMNAPPM1BPTPN1PPP1CCTSHR
SCHEMBL2139493 0.68 LMNA (0.40) LMNAPOLBPPM1BPTPN1PPP1CC
SCHEMBL21076384 0.67 PPM1B (0.36) PPM1BPTPN1PPP1CCKDM4ETSHR
SCHEMBL14966710 0.66 SOAT1 (0.39) LMNAPOLBPPM1BPTPN1PPP1CC
SCHEMBL14967349 0.66 PPM1B (0.42) LMNAPOLBPPM1BPTPN1PPP1CC
SCHEMBL18166928 0.64 ALDH1A1 (0.37) LMNAPPM1BPTPN1PPP1CCKDM4E
SCHEMBL4157000 0.63 LMNA (0.60) LMNAPPM1BPTPN1PPP1CCKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821668-B1 DERIVATIVES OF SUCCINAMIDE AND THEIR USE AS METALLOPROTEINASE INHIBITOR BRITISH BIOTECH PHARM (GB) 2000-08-23 EP disclosed
US-5908851-A TUMOR NECROSIS FACTOR, COLLAGENASE, STROMELYSIN, AND GELATINASE INHIBITORS; OSTEOPOROSIS, RHEUMATIC AND ORAL DISEASES; ANTIARTHRITIC AND ANTIULCER AGENTS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1999-06-01 US disclosed
EP-0821668-A1 DERIVATIVES OF SUCCINAMIDE AND THEIR USE AS METALLOPROTEINASE INHIBITOR BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1998-02-04 EP disclosed
WO-1996033165-A1 DERIVATIVES OF SUCCINAMIDE AND THEIR USE AS METALLOPROTEINASE INHIBITOR BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1996-10-24 WO disclosed