SCHEMBL8076789

SCHEMBL8076789

CC(=O)N(Cc1ccccc1)c1ccc(C(=O)CSc2ccnc3ccccc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 3/20 0.46
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
TSPO P30536 1/20 0.41
HPGD P15428 2/20 0.41
CYP2C19 P33261 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 2/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ALDH1A1 P00352 6/20 0.39
MAPT P10636 4/20 0.39
CYP2C9 P11712 1/20 0.39
MAOB P27338 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
POLB P06746 1/20 0.39
HSP90AA1 P07900 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084097 0.82 HTR2C (0.48) KMT2AMEN1HPGDCYP2C19CYP3A4
SCHEMBL8084102 0.81 HTR2C (0.53) KMT2AMEN1HPGDCYP2C19CYP3A4
SCHEMBL8090035 0.78 SMN1; SMN2 (0.54) HPGDCYP2C19CYP3A4CYP1A2HIF1A
SCHEMBL8088268 0.78 HSD17B10 (0.50) KMT2AMEN1HPGDCYP2C19CYP3A4
SCHEMBL8076734 0.77 HDAC6 (0.47) KMT2AMEN1HPGDCYP2C19CYP3A4
SCHEMBL8084739 0.76 ALDH1A1 (0.60) KMT2AMEN1HPGDCYP2C19CYP3A4
SCHEMBL8084757 0.76 ALDH1A1 (0.49) KMT2AMEN1HPGDCYP2C19CYP3A4
SCHEMBL8084741 0.76 ALDH1A1 (0.50) KMT2AMEN1HPGDCYP2C19CYP3A4
SCHEMBL8076747 0.73 CYP1A2 (0.55) KMT2AMEN1HPGDCYP1A2ALDH1A1
SCHEMBL8084836 0.72 ALDH1A1 (0.54) KMT2AMEN1HPGDCYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057447-A BACTERICIDES FOR CAMPYLOBACTER ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2000-05-02 US disclosed
EP-0926139-A1 QUINOLINE SULFIDE DERIVATIVES ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 1999-06-30 EP disclosed