SCHEMBL8084097

SCHEMBL8084097

CN(C)c1ccc(C(=O)CSc2ccnc3ccccc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
CNR2 P34972 1/20 0.46
HPGD P15428 3/20 0.44
CYP2C19 P33261 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 1/20 0.43
HIF1A Q16665 1/20 0.43
ALDH1A1 P00352 8/20 0.43
MAPT P10636 5/20 0.43
CYP2C9 P11712 1/20 0.43
MAOB P27338 1/20 0.43
KMT2A Q03164 4/20 0.42
MEN1 O00255 2/20 0.42
KDM4E B2RXH2 5/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
ALOX15 P16050 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084102 0.88 HTR2C (0.53) HTR2CHTR2BHPGDCYP2C19HSD17B10
SCHEMBL8088268 0.85 HSD17B10 (0.50) HPGDCYP2C19HSD17B10CYP1A2CYP3A4
SCHEMBL8084741 0.83 ALDH1A1 (0.50) HPGDCYP2C19HSD17B10CYP1A2CYP3A4
SCHEMBL8084739 0.83 ALDH1A1 (0.60) HPGDCYP2C19HSD17B10CYP1A2CYP3A4
SCHEMBL8076789 0.82 PDK1 (0.46) HPGDCYP2C19HSD17B10CYP1A2CYP3A4
SCHEMBL8084757 0.81 ALDH1A1 (0.49) HPGDCYP2C19HSD17B10CYP1A2CYP3A4
SCHEMBL8076747 0.80 CYP1A2 (0.55) HPGDCYP1A2ALDH1A1MAPTKMT2A
SCHEMBL8084836 0.79 ALDH1A1 (0.54) HPGDCYP2C19HSD17B10CYP1A2CYP3A4
SCHEMBL8088227 0.78 DNMT1 (0.44) HTR2CHTR2BHPGDHSD17B10ALDH1A1
SCHEMBL8084734 0.78 HTR2C (0.44) HTR2CHTR2BCNR2HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057447-A BACTERICIDES FOR CAMPYLOBACTER ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 2000-05-02 US disclosed
EP-0926139-A1 QUINOLINE SULFIDE DERIVATIVES ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 1999-06-30 EP disclosed