SCHEMBL20343752

SCHEMBL20343752

Nc1nc(-c2cncnc2)nc2c1NCN2Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.39
ADORA3 P0DMS8 3/20 0.39
ADORA1 P30542 3/20 0.37
DHPS P49366 3/20 0.36
GBA1 P04062 2/20 0.35
TLR7 Q9NYK1 1/20 0.35
MAPK1 P28482 1/20 0.35
LMNA P02545 1/20 0.33
ACHE P22303 1/20 0.33
CFTR P13569 3/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14944658 0.76 TLR7 (0.36) ADORA2AADORA3ADORA1TLR7MAPK1
SCHEMBL28852897 0.75 HSP90AA1 (0.40) TLR7LMNA
SCHEMBL14944653 0.74 DRD2 (0.31) ADORA2AADORA3MAPK1
SCHEMBL14944729 0.74 ALDH1A1 (0.32) ADORA2AADORA3TLR7
SCHEMBL14944685 0.73 TLR7 (0.33) TLR7
SCHEMBL14944688 0.72 ALDH1A1 (0.30)
SCHEMBL19423858 0.71 CCR5 (0.31) TLR7
SCHEMBL4144591 0.69 HPRT1 (0.50)
SCHEMBL28184098 0.69 MAPK1 (0.39) TLR7MAPK1
SCHEMBL28183208 0.69 ABCB1 (0.38) TLR7LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776439-B1 PURINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS JANSSEN SCIENCES IRELAND UC (IE) 2018-07-04 EP disclosed