SCHEMBL8077310

SCHEMBL8077310

CC(=O)Nc1cc(Br)cn(C2=CC(C)(C)Oc3ccc(C#N)cc32)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
KDM4E B2RXH2 1/20 0.34
GPR35 Q9HC97 1/20 0.31
ABCC9 O60706 5/20 0.31
DRD2 P14416 3/20 0.31
DRD3 P35462 3/20 0.31
KCNE1 P15382 3/20 0.31
KCNQ1 P51787 3/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
KCND3 Q9UK17 1/20 0.31
DYRK1A Q13627 1/20 0.30
ABCB1 P08183 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088696 0.89 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL8085352 0.85 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL8090750 0.85 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL8085129 0.84 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL8084934 0.83 CFTR (0.38) KDM4ECYP1A2KMT2ADYRK1A
SCHEMBL8084925 0.83 EGLN2 (0.33) KDM4EGPR35ABCC9DRD2DRD3
SCHEMBL9378613 0.83 ABCC9 (0.33) KDM4EGPR35ABCC9DRD2DRD3
SCHEMBL8077281 0.82 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL8090684 0.81 EGLN2 (0.38) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL9733641 0.81 OTUD7B (0.31) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed