SCHEMBL8085352

SCHEMBL8085352

CC(=O)Nc1cc(Br)c(=O)n(C2=CC(C)(C)Oc3ccc(C#N)cc32)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
DRD2 P14416 6/20 0.36
DRD3 P35462 6/20 0.36
KDM4E B2RXH2 1/20 0.34
EGLN2 Q96KS0 4/20 0.33
ABCC9 O60706 5/20 0.33
ABCC8 Q09428 2/20 0.32
KCNJ11 Q14654 2/20 0.32
KCNJ8 Q15842 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 1/20 0.32
KDM1A O60341 1/20 0.31
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090684 0.89 EGLN2 (0.38) PDE4APDE4BPDE4CPDE4DDRD2
SCHEMBL8088372 0.87 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DDRD2
SCHEMBL8077310 0.85 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DDRD2
SCHEMBL8085129 0.84 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL8090476 0.83 SMN1; SMN2 (0.38) KDM4ECYP1A2
SCHEMBL8077023 0.83 EGLN2 (0.36) DRD2DRD3KDM4EEGLN2ABCC9
SCHEMBL9376786 0.83 DRD2 (0.37) DRD2DRD3KDM4EEGLN2ABCC9
SCHEMBL8084279 0.82 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL8088696 0.81 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DDRD2
SCHEMBL9733537 0.81 EGLN2 (0.33) DRD2DRD3EGLN2CYP1A2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed