SCHEMBL8085347

SCHEMBL8085347

COc1cccn(C2=C(C)C(C)(C)Oc3ccc([N+](=O)[O-])cc32)c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
MAPT P10636 6/20 0.35
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
RECQL P46063 1/20 0.34
DUSP3 P51452 1/20 0.34
PTPN5 P54829 1/20 0.34
PTPN11 Q06124 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
NPC1 O15118 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088675 0.89 RECQL (0.44) HTTTDP1MAPTALDH1A1SMN1; SMN2
SCHEMBL8077334 0.86 ALDH1A1 (0.38) TDP1MAPTALDH1A1KMT2AMEN1
SCHEMBL8076907 0.85 TDP1 (0.37) HTTTDP1ALDH1A1KMT2AMEN1
SCHEMBL8084426 0.85 ALDH1A1 (0.36) TDP1ALDH1A1KMT2AMEN1CYP3A4
SCHEMBL8077303 0.85 ALDH1A1 (0.36) TDP1ALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL8090492 0.83 KDM4E (0.36) HTTTDP1MAPTALDH1A1KMT2A
SCHEMBL8085346 0.82 ALDH1A1 (0.38) TDP1MAPTALDH1A1KMT2AMEN1
SCHEMBL8090777 0.82 PDE4A (0.38) KMT2AMEN1
SCHEMBL8085103 0.81 CFTR (0.41) HTTMAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL8088445 0.80 ADORA3 (0.41) ADORA3ADORA2AHTTTDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed