SCHEMBL8081670

SCHEMBL8081670

Nc1cc(Br)ccc1Oc1ccccc1C(=O)OC(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
POLB P06746 3/20 0.39
MAPT P10636 2/20 0.39
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
GLA P06280 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GAA P10253 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CTNNB1 P35222 1/20 0.35
HTT P42858 2/20 0.34
SLC6A3 Q01959 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LRRK2 Q5S007 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8075178 0.86 ALDH1A1 (0.46) KDM4ELMNAALDH1A1HPGDMAPT
SCHEMBL8067090 0.85 SLC6A4 (0.44) KDM4ELMNAALDH1A1HPGDMAPT
SCHEMBL5720159 0.82 MAPT (0.43) KDM4ELMNAALDH1A1HPGDPOLB
SCHEMBL8067203 0.82 KDM4E (0.51) KDM4ELMNAALDH1A1HPGDPOLB
Diphenylmethanol SCHEMBL8081675 0.81 HTT (0.43) KDM4ELMNAALDH1A1HPGDPOLB
SCHEMBL8080271 0.73 CCR2 (0.52) KDM4EGAA
SCHEMBL13261645 0.73 NCOA1 (0.50) LMNAALDH1A1POLBMAPTPTGDR2
SCHEMBL28058117 0.72 ESR1 (0.61) KDM4ELMNAALDH1A1HPGDPOLB
SCHEMBL8076970 0.70 L3MBTL1 (0.52) KDM4ELMNAALDH1A1HPGDMAPT
SCHEMBL8081645 0.69 L3MBTL1 (0.43) KDM4ELMNAALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799198-B1 ANTI-INFLAMMATORY COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2000-08-30 EP disclosed
EP-0799198-A4 1997-10-15 EP disclosed
EP-0799198-A1 ANTI-INFLAMMATORY COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1997-10-08 EP disclosed
US-5545669-A Anti-inflammatory compounds SMITHKLINE BEECHAM CORPORATION 1996-08-13 US disclosed
WO-1995033461-A1 ANTI-INFLAMMATORY COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-14 WO disclosed