SCHEMBL8082470

SCHEMBL8082470

CC1=C(C(=O)OC(C)C)C(c2cccc(Cl)c2Cl)C2=C(N1)C(=O)OC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.51
CYP2C9 P11712 5/20 0.47
CYP1A2 P05177 4/20 0.47
CYP3A4 P08684 4/20 0.47
CYP2C19 P33261 4/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
KDM4E B2RXH2 3/20 0.47
ABCB11 O95342 3/20 0.47
MAPT P10636 3/20 0.47
HIF1A Q16665 2/20 0.47
HSD17B10 Q99714 2/20 0.47
TSHR P16473 2/20 0.47
CYP2D6 P10635 2/20 0.47
NR1I2 O75469 2/20 0.47
NR3C1 P04150 2/20 0.47
ADORA3 P0DMS8 2/20 0.47
TBXA2R P21731 2/20 0.47
OPRK1 P41145 2/20 0.47
SLC6A3 Q01959 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047294 0.85 ALOX15 (0.40) ALOX15CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7984491 0.82 ABCC1 (0.48) ALOX15MEN1KMT2AKDM4EMAPT
SCHEMBL8086984 0.79 PYGL (0.45) ALOX15ALDH1A1LMNAPOLBADORA2B
SCHEMBL7273889 0.79 CYP2C9 (0.60) ALOX15CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7408943 0.79 CYP2C9 (0.73) ALOX15CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL29664498 0.79 CYP2C9 (0.60) ALOX15CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7981102 0.75 HSD17B10 (0.64) ALOX15MEN1KMT2AKDM4EMAPT
SCHEMBL7979577 0.74 KDM4E (0.62) ALOX15KDM4EHSD17B10TSHRNPSR1
SCHEMBL7410229 0.74 CYP2C9 (0.66) ALOX15CYP2C9CYP1A2CYP3A4CYP2C19
SCHEMBL7429254 0.73 CYP2C9 (0.64) ALOX15CYP2C9CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121284-A SPECIFIED 1-(ALKYL OR CYCLOALKYL)-2-METHYL-3-(ALKOXYCARBONYL)-4-(SUBSTITUTED PYRIDYL OR ARYL)-5-OXO-1,4,5,6,7,8-HEXAHYDROQUINOLINE COMPOUNDS; TREATING SICKLE CELL ANEMIA, PSYCHOSES, DEPRESSION BAYER AKTIENGESELLSCHAFT (DE) 2000-09-19 US disclosed