SCHEMBL8083504

SCHEMBL8083504

COc1c(CCCc2cccnc2)[c]c(-c2cccnc2)c(OC)c1OC

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP2A6 P11509 1/20 0.41
PTAFR P25105 6/20 0.40
HRH1 P35367 2/20 0.40
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CHRNA7 P36544 2/20 0.38
TBXAS1 P24557 4/20 0.37
GPR84 Q9NQS5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5834366 0.94 CYP11B1 (0.42) TDP1L3MBTL1GPR84
SCHEMBL8095186 0.88 TDP1 (0.51) TDP1L3MBTL1CYP2A6PTAFRHRH1
SCHEMBL8091559 0.85 TDP1 (0.48) TDP1L3MBTL1CYP2A6PTAFRHRH1
SCHEMBL8091379 0.80 HTR2A (0.35) TDP1L3MBTL1
SCHEMBL8098200 0.74 HTT (0.43) CYP2A6
SCHEMBL8827622 0.74 CYP11B1 (0.42) TDP1L3MBTL1GPR84
SCHEMBL8083417 0.72 PRKCI (0.34)
SCHEMBL8083550 0.71 KDM4E (0.38)
SCHEMBL7430378 0.71 L3MBTL1 (0.38) L3MBTL1
SCHEMBL6567905 0.71 HTR2A (0.41) TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124328-A TREATING NERVE CELLS WITH A NEUROTROPHIC AGENT; PROMOTING REPAIR OF NEURONAL DAMAGE CAUSED BY DISEASE OR PHYSICAL TRAUMA VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-09-26 US disclosed
US-6037370-A TREATING ALZHEIMER*S DISEASE, AMYOTROPHIC LATERAL SCLEROSIS, PARKINSON*S DISEASE, AND OTHER NERVOUS SYSTEM DISORDERS WITH PEPTIDE DERIVATIVES VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-03-14 US disclosed