SCHEMBL8091559

SCHEMBL8091559

COc1c(CCCc2ccccc2)[c]c(CCCc2cccnc2)c(OC)c1OC

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CYP2A6 P11509 1/20 0.45
TBXAS1 P24557 7/20 0.43
HRH1 P35367 2/20 0.43
HRH4 Q9H3N8 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
CHRNA7 P36544 3/20 0.41
PTAFR P25105 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095186 0.96 TDP1 (0.51) TDP1L3MBTL1CYP2A6TBXAS1HRH1
SCHEMBL6567905 0.87 HTR2A (0.41) TDP1L3MBTL1
SCHEMBL7430378 0.85 L3MBTL1 (0.38) L3MBTL1
SCHEMBL8083504 0.85 TDP1 (0.43) TDP1L3MBTL1CYP2A6TBXAS1HRH1
SCHEMBL8091400 0.84 L3MBTL1 (0.44) TDP1L3MBTL1
SCHEMBL8090038 0.84 ABCB1 (0.39) TDP1L3MBTL1
SCHEMBL8090053 0.81 LTA4H (0.40) L3MBTL1
SCHEMBL7434046 0.80 TDP1 (0.51) TDP1L3MBTL1
SCHEMBL7428315 0.80 KDM4E (0.41) TDP1HRH1HRH4HRH3
SCHEMBL8200325 0.79 CYP2A6 (0.68) TDP1L3MBTL1CYP2A6TBXAS1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124328-A TREATING NERVE CELLS WITH A NEUROTROPHIC AGENT; PROMOTING REPAIR OF NEURONAL DAMAGE CAUSED BY DISEASE OR PHYSICAL TRAUMA VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-09-26 US disclosed
US-6037370-A TREATING ALZHEIMER*S DISEASE, AMYOTROPHIC LATERAL SCLEROSIS, PARKINSON*S DISEASE, AND OTHER NERVOUS SYSTEM DISORDERS WITH PEPTIDE DERIVATIVES VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-03-14 US disclosed