SCHEMBL8091379

SCHEMBL8091379

COc1c(CCCc2ccccc2)[c]c(-c2ccccc2)c(OC)c1OC

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8827644 0.91 BCHE (0.42)
SCHEMBL6567905 0.88 HTR2A (0.41) HTR2AL3MBTL1TDP1IDO1
SCHEMBL8083417 0.87 PRKCI (0.34) HTR2A
SCHEMBL8083550 0.86 KDM4E (0.38) ALDH1A1
SCHEMBL8090038 0.84 ABCB1 (0.39) HTR2AL3MBTL1TDP1IDO1
SCHEMBL8091400 0.84 L3MBTL1 (0.44) L3MBTL1TDP1
SCHEMBL8090053 0.82 LTA4H (0.40) HTR2AL3MBTL1
SCHEMBL7434046 0.81 TDP1 (0.51) L3MBTL1TDP1ALDH1A1
SCHEMBL8083504 0.80 TDP1 (0.43) L3MBTL1TDP1
SCHEMBL8090170 0.78 TDP1 (0.49) L3MBTL1TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124328-A TREATING NERVE CELLS WITH A NEUROTROPHIC AGENT; PROMOTING REPAIR OF NEURONAL DAMAGE CAUSED BY DISEASE OR PHYSICAL TRAUMA VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-09-26 US disclosed
US-6037370-A TREATING ALZHEIMER*S DISEASE, AMYOTROPHIC LATERAL SCLEROSIS, PARKINSON*S DISEASE, AND OTHER NERVOUS SYSTEM DISORDERS WITH PEPTIDE DERIVATIVES VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-03-14 US disclosed