SCHEMBL8084547

SCHEMBL8084547

CC1=C(n2c(Cl)cccc2=O)c2cc([N+](=O)[O-])ccc2OC1(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
MALT1 Q9UDY8 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 1/20 0.34
ATM Q13315 1/20 0.34
PTPRC P08575 3/20 0.33
S100A4 P26447 2/20 0.33
ACHE P22303 2/20 0.33
CASP1 P29466 1/20 0.33
CASP3 P42574 1/20 0.33
CASP4 P49662 1/20 0.33
CASP7 P55210 1/20 0.33
CASP9 P55211 1/20 0.33
CASP6 P55212 1/20 0.33
TSHR P16473 1/20 0.33
BCHE P06276 1/20 0.33
CES1 P23141 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
BCL2A1 Q16548 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090782 0.80 ABCC9 (0.36) MALT1CASP3
SCHEMBL8085346 0.80 ALDH1A1 (0.38) ALDH1A1MALT1TDP1CYP3A4PTPRC
SCHEMBL8084294 0.79 ALDH1A1 (0.37) ALDH1A1MALT1TDP1CYP3A4ATM
SCHEMBL8085089 0.78 MEN1 (0.37) ALDH1A1MALT1TDP1CYP3A4PTPRC
SCHEMBL8077303 0.77 ALDH1A1 (0.36) ALDH1A1MALT1TDP1CYP3A4PTPRC
SCHEMBL8085417 0.77 MALT1 (0.37) ALDH1A1MALT1TDP1CYP3A4PTPRC
SCHEMBL8084975 0.76 HSD17B10 (0.37) ALDH1A1MALT1TDP1CYP3A4PTPRC
SCHEMBL8077012 0.75 MEN1 (0.36) ALDH1A1MALT1TDP1CYP3A4PTPRC
SCHEMBL8084565 0.74 MEN1 (0.36) ALDH1A1MALT1TDP1CYP3A4PTPRC
SCHEMBL8077334 0.74 ALDH1A1 (0.38) ALDH1A1MALT1TDP1CYP3A4PTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed