SCHEMBL8084591

SCHEMBL8084591

O=C(CCCCc1ccc(Cl)c(Cl)c1)N1CCC(c2ccc(Cl)cc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 5/20 0.48
GRM5 P41594 1/20 0.47
CCR2 P41597 2/20 0.47
KCNH2 Q12809 1/20 0.47
NAAA Q02083 1/20 0.46
CCR1 P32246 1/20 0.45
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
CACNA1G O43497 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092580 0.91 GRM5 (0.53) MCHR1GRM5NAAACCR1KMT2A
SCHEMBL8091484 0.85 DRD2 (0.55) MCHR1GRM5NAAACCR1KMT2A
SCHEMBL8091568 0.85 MEN1 (0.54) CCR1KMT2AMEN1ALDH1A1LMNA
SCHEMBL3878560 0.81 CCR1 (0.58) GRM5CCR1KMT2AMEN1CACNA1G
SCHEMBL3869863 0.80 MCHR1 (0.54) MCHR1GRM5CCR1KMT2AMEN1
SCHEMBL8097197 0.80 NAAA (0.55) NAAACCR1KMT2AMEN1ALDH1A1
SCHEMBL3870960 0.78 CCR1 (0.50) MCHR1GRM5CCR1KMT2AMEN1
SCHEMBL3867771 0.78 CCR1 (0.50) MCHR1GRM5CCR1KMT2AMEN1
SCHEMBL3994513 0.76 MAPT (0.53) MCHR1KMT2AMEN1ALDH1A1LMNA
SCHEMBL30616890 0.76 MCHR1 (0.44) MCHR1GRM5NAAACCR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US claimed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP claimed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO claimed