SCHEMBL8091568

SCHEMBL8091568

O=C(CCCCc1ccc(Cl)cc1)N1CCC(c2ccccc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
HSD11B1 P28845 1/20 0.53
IDO1 P14902 1/20 0.52
CCR1 P32246 4/20 0.52
MAPT P10636 3/20 0.51
TP53 P04637 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
CACNA1G O43497 2/20 0.49
CACNA1H O95180 1/20 0.49
LMNA P02545 2/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
MAPK1 P28482 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092580 0.94 GRM5 (0.53) MEN1KMT2ACCR1LMNAALDH1A1
SCHEMBL3878560 0.91 CCR1 (0.58) MEN1KMT2AHSD11B1CCR1MAPT
SCHEMBL8092824 0.91 SIGMAR1 (0.59) MEN1KMT2AMAPTTP53CYP1A2
SCHEMBL8091484 0.88 DRD2 (0.55) MEN1KMT2ACCR1
SCHEMBL9377300 0.88 DRD2 (0.53) MEN1KMT2AMAPTTP53CYP1A2
SCHEMBL8097197 0.87 NAAA (0.55) MEN1KMT2ACCR1MAPTTP53
SCHEMBL8092966 0.85 ALDH1A1 (0.64) KMT2AHSD11B1MAPTTSHRSIGMAR1
SCHEMBL8084591 0.85 MCHR1 (0.48) MEN1KMT2ACCR1CACNA1GLMNA
SCHEMBL3869863 0.82 MCHR1 (0.54) MEN1KMT2ACCR1LMNAALDH1A1
SCHEMBL3867771 0.81 CCR1 (0.50) MEN1KMT2ACCR1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP claimed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO claimed
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed