SCHEMBL8084594

SCHEMBL8084594

FC(F)(F)c1ccc(-c2ncc(-c3ccc(Br)cc3)s2)cc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.57
TRPV1 Q8NER1 1/20 0.49
SNCA P37840 2/20 0.43
HSD17B1 P14061 3/20 0.43
HSD17B2 P37059 3/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HDAC6 Q9UBN7 3/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC4 P56524 1/20 0.38
KIF11 P52732 1/20 0.38
AHR P35869 1/20 0.38
CDK2 P24941 3/20 0.36
AKT1 P31749 3/20 0.36
PTPN1 P18031 1/20 0.36
PRMT5 O14744 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30279827 0.92 HSD17B1 (0.49) XDHSNCAHSD17B1HSD17B2CYP3A4
SCHEMBL13191551 0.87 HSD17B1 (0.46) XDHTRPV1SNCAHSD17B1HSD17B2
SCHEMBL18167775 0.87 KIF11 (0.45) XDHSNCAHSD17B1HSD17B2CYP3A4
SCHEMBL7218452 0.80 CSNK2A1 (0.55) HDAC6HDAC1HDAC4
SCHEMBL8085528 0.80 GCK (0.45) XDHHSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL13494529 0.79 MAPT (0.44) HSD17B1HSD17B2CYP3A4CYP2C9KIF11
SCHEMBL10630306 0.77 GCK (0.39) HSD17B1HSD17B2CYP3A4CYP2C9KIF11
SCHEMBL21484979 0.77 KIF11 (0.41) SNCAHSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL10464166 0.77 TP53 (0.42) HSD17B1HSD17B2CYP3A4CYP2C9KIF11
SCHEMBL3057473 0.75 KIF11 (0.44) TRPV1HDAC6HDAC1KIF11CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6011048-A Thiazole benzenesulfonamides as β3 agonists for treatment of diabetes and obesity MERCK & CO., INC. (US) 2000-01-04 US disclosed