SCHEMBL8085528

SCHEMBL8085528

O=S(=O)(Cl)c1ccc(-c2cnc(-c3ccc(C(F)(F)F)cc3)s2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCK P35557 2/20 0.45
GCKR Q14397 2/20 0.45
KIF11 P52732 2/20 0.43
XDH P47989 1/20 0.43
MLYCD O95822 1/20 0.40
MMP2 P08253 3/20 0.40
MMP9 P14780 3/20 0.40
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
HSD17B1 P14061 2/20 0.39
HSD17B2 P37059 2/20 0.39
HDAC6 Q9UBN7 2/20 0.38
HDAC1 Q13547 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8193542 0.87 HSD17B1 (0.48) MMP2MMP9CYP3A4CYP2C9HSD17B1
SCHEMBL30279827 0.87 HSD17B1 (0.49) KIF11XDHCYP3A4CYP2C9HSD17B1
SCHEMBL18167775 0.82 KIF11 (0.45) GCKGCKRKIF11XDHCYP3A4
SCHEMBL13191551 0.82 HSD17B1 (0.46) KIF11XDHCYP3A4CYP2C9HSD17B1
SCHEMBL8084594 0.80 XDH (0.57) KIF11XDHCYP3A4CYP2C9HSD17B1
SCHEMBL3071920 0.78 KIF11 (0.66) KIF11MMP2MMP9KDM1APTGS2
SCHEMBL7218452 0.78 CSNK2A1 (0.55) HDAC6HDAC1KDM4EALDH1A1HDAC4
SCHEMBL61336 0.76 KIF11 (0.55) KIF11ALDH1A1MAPTPTGS2CA1
SCHEMBL13494529 0.75 MAPT (0.44) KIF11CYP3A4CYP2C9HSD17B1HSD17B2
SCHEMBL10464166 0.72 TP53 (0.42) KIF11CYP3A4CYP2C9HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6011048-A Thiazole benzenesulfonamides as β3 agonists for treatment of diabetes and obesity MERCK & CO., INC. (US) 2000-01-04 US disclosed