SCHEMBL8084693

SCHEMBL8084693

O=C(/C=C/C(=O)OC1=NC(Cc2ccc3ccccc3c2)CN1)OC1=NC(Cc2ccc3ccccc3c2)CN1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.36
SLC6A4 P31645 7/20 0.36
KCNH2 Q12809 3/20 0.36
SLC6A3 Q01959 6/20 0.36
CYP2D6 P10635 1/20 0.35
NFKB1 P19838 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
TBXA2R P21731 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGFR P43088 1/20 0.35
PTGER3 P43115 1/20 0.35
PTGER2 P43116 1/20 0.35
PTGDR Q13258 1/20 0.35
CCNB2 O95067 1/20 0.35
CCNE2 O96020 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNA2 P20248 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093566 0.85 ADRA2A (0.46)
SCHEMBL8091875 0.71 ADRA2A (0.43) SLC6A2SLC6A4SLC6A3HTR2AHTR2C
SCHEMBL8085006 0.71 ADRA2A (0.43) SLC6A2SLC6A4SLC6A3HTR2AHTR2C
SCHEMBL27500912 0.71 MMP13 (0.35) KCNH2CYP2D6TBXA2RPTGER4PTGFR
Fumaric Acid SCHEMBL8084690 0.70 TBXA2R (0.43) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
Fumaric Acid SCHEMBL8084695 0.70 TBXA2R (0.43) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL11821505 0.67 SLC6A4 (0.49) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL8084748 0.67 CYP11B2 (0.39)
SCHEMBL8090880 0.66 MCHR1 (0.32)
SCHEMBL8093366 0.66 ADRA2A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127396-A Imidazoline compounds ADIR ET COMPAGNIE (FR) 2000-10-03 US disclosed