SCHEMBL8085153

SCHEMBL8085153

CC1(C)C=C(n2cc(Br)cc([N+](=O)[O-])c2=O)c2cc(C#N)ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
ABCC9 O60706 1/20 0.37
VCAM1 P19320 1/20 0.34
GPR35 Q9HC97 1/20 0.33
MAPT P10636 1/20 0.31
AR P10275 1/20 0.30
MALT1 Q9UDY8 1/20 0.30
P2RY6 Q15077 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088704 0.90 ABCC9 (0.40) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8085300 0.89 VCAM1 (0.39) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8085257 0.87 MEN1 (0.34) ARMALT1
SCHEMBL8085129 0.86 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8085433 0.85 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL7277069 0.84 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8077281 0.84 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8077169 0.82 ABCC9 (0.36) ABCC9VCAM1GPR35MAPTAR
SCHEMBL9372285 0.82 ABCC9 (0.36) ABCC9VCAM1GPR35MAPTAR
SCHEMBL8085246 0.82 ABCC9 (0.39) PDE4APDE4BPDE4CPDE4DABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed