SCHEMBL8085300

SCHEMBL8085300

CC1(C)C=C(n2cc(Cl)cc([N+](=O)[O-])c2=O)c2cc(C#N)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 3/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
ABCC9 O60706 6/20 0.37
P2RY6 Q15077 1/20 0.32
MERTK Q12866 2/20 0.31
MAPT P10636 1/20 0.31
AR P10275 1/20 0.30
MALT1 Q9UDY8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088704 0.90 ABCC9 (0.40) VCAM1PDE4APDE4BPDE4CPDE4D
SCHEMBL8085153 0.89 PDE4A (0.38) VCAM1PDE4APDE4BPDE4CPDE4D
SCHEMBL8089644 0.87 MEN1 (0.34) MAPTMALT1
SCHEMBL8085358 0.86 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8085246 0.85 ABCC9 (0.39) VCAM1PDE4APDE4BPDE4CPDE4D
SCHEMBL7277069 0.84 PDE4A (0.39) VCAM1PDE4APDE4BPDE4CPDE4D
SCHEMBL8077016 0.84 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8084273 0.82 VCAM1 (0.38) VCAM1ABCC9P2RY6MERTKMAPT
SCHEMBL9372978 0.82 VCAM1 (0.38) VCAM1ABCC9P2RY6MERTKMAPT
SCHEMBL8085433 0.82 PDE4A (0.40) VCAM1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed