SCHEMBL7277069

SCHEMBL7277069

CC1(C)C=C(n2cccc([N+](=O)[O-])c2=O)c2cc(C#N)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
ABCC9 O60706 7/20 0.38
VCAM1 P19320 1/20 0.35
MAPT P10636 4/20 0.34
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
AR P10275 1/20 0.31
PTPN1 P18031 1/20 0.31
ABCC8 Q09428 1/20 0.31
KCNJ11 Q14654 1/20 0.31
KCNJ8 Q15842 1/20 0.31
MALT1 Q9UDY8 1/20 0.31
P2RY6 Q15077 1/20 0.31
ABCB1 P08183 2/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090699 0.86 ALDH1A1 (0.37) MAPTPOLBMAPK1TDP1MALT1
SCHEMBL8088704 0.86 ABCC9 (0.40) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8085300 0.84 VCAM1 (0.39) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8085153 0.84 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8090271 0.83 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL7277201 0.83 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL8088878 0.83 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL7267332 0.83 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9299309 0.83 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9372282 0.82 ABCC9 (0.38) ABCC9VCAM1MAPTPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0346724-A1 Chroman derivates MERCK PATENT GmbH (DE) 1989-12-20 EP disclosed