SCHEMBL8085331

SCHEMBL8085331

CC1(C)C=C(n2cc([N+](=O)[O-])cc(Cl)c2=O)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.38
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PTPRC P08575 1/20 0.34
S100A4 P26447 1/20 0.34
CASP3 P42574 2/20 0.34
CASP1 P29466 1/20 0.34
CASP4 P49662 1/20 0.34
CASP7 P55210 1/20 0.34
CASP9 P55211 1/20 0.34
CASP6 P55212 1/20 0.34
KMT2A Q03164 2/20 0.33
MALT1 Q9UDY8 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084998 0.92 ALDH1A1 (0.34) HSD17B10ALDH1A1CYP3A4TDP1PTPRC
SCHEMBL8088693 0.90 PDE7A (0.33) HSD17B10ALDH1A1CYP3A4TDP1PTPRC
SCHEMBL8085246 0.88 ABCC9 (0.39) MALT1
SCHEMBL8085338 0.88 KMT2A (0.38) ALDH1A1CYP3A4TDP1PTPRCS100A4
SCHEMBL8084409 0.87 ALDH1A1 (0.35) ALDH1A1CYP3A4TDP1PTPRCS100A4
SCHEMBL8085305 0.86 ALDH1A1 (0.36) HSD17B10ALDH1A1CYP3A4TDP1PTPRC
SCHEMBL8088667 0.85 KMT2A (0.42) ALDH1A1CYP3A4KMT2ALMNAMEN1
SCHEMBL7300724 0.85 PDE4B (0.32) ALDH1A1KMT2AMEN1MAPT
SCHEMBL8089644 0.85 MEN1 (0.34) ALDH1A1CYP3A4TDP1PTPRCS100A4
SCHEMBL8084458 0.84 TDP1 (0.34) ALDH1A1CYP3A4TDP1PTPRCS100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed