SCHEMBL8085338

SCHEMBL8085338

CC1(C)C=C(n2cc([N+](=O)[O-])cc([N+](=O)[O-])c2=O)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.38
MEN1 O00255 4/20 0.38
ADORA2B P29275 1/20 0.35
ALDH1A1 P00352 4/20 0.35
TDP1 Q9NUW8 3/20 0.35
CYP3A4 P08684 1/20 0.35
PTPRC P08575 1/20 0.35
S100A4 P26447 1/20 0.35
CASP3 P42574 2/20 0.34
CASP1 P29466 1/20 0.34
CASP4 P49662 1/20 0.34
CASP7 P55210 1/20 0.34
CASP9 P55211 1/20 0.34
CASP6 P55212 1/20 0.34
MAPK1 P28482 2/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GPR35 Q9HC97 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085257 0.90 MEN1 (0.34) KMT2AMEN1ADORA2BALDH1A1TDP1
SCHEMBL8089644 0.90 MEN1 (0.34) KMT2AMEN1ADORA2BALDH1A1TDP1
SCHEMBL8084409 0.88 ALDH1A1 (0.35) KMT2AMEN1ALDH1A1TDP1CYP3A4
SCHEMBL8085331 0.88 HSD17B10 (0.38) KMT2AMEN1ALDH1A1TDP1CYP3A4
SCHEMBL8088704 0.87 ABCC9 (0.40) KMT2AMEN1TDP1MAPK1MALT1
SCHEMBL8206417 0.87 MEN1 (0.35) KMT2AMEN1ADORA2BALDH1A1TDP1
SCHEMBL8090699 0.85 ALDH1A1 (0.37) KMT2AMEN1ADORA2BALDH1A1TDP1
SCHEMBL7291279 0.85 ADORA2B (0.31) KMT2AMEN1ADORA2BALDH1A1MAPT
SCHEMBL8085035 0.85 ALDH1A1 (0.38) KMT2AMEN1ALDH1A1TDP1CYP3A4
SCHEMBL7291070 0.84 CCNC (0.35) KMT2AMEN1ADORA2BALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed