SCHEMBL8085342

SCHEMBL8085342

COC(=O)c1ccc2c(c1)C(n1ccccc1=O)C(C)(O)C(C)(C)O2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.39
PDK2 Q15119 2/20 0.33
NPC1 O15118 2/20 0.33
IDH1 O75874 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
FGFR1 P11362 1/20 0.33
TRPA1 O75762 1/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
NPY5R Q15761 1/20 0.33
ALOX15 P16050 2/20 0.32
RBP4 P02753 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PARP1 P09874 1/20 0.32
IDO1 P14902 1/20 0.32
FBP1 P09467 1/20 0.32
EDNRA P25101 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090564 0.89 MAPT (0.41) RAB9ASMN1; SMN2ALDH1A1LMNACA12
SCHEMBL8088411 0.88 KDM4E (0.33) ALDH1A1
SCHEMBL8088453 0.87 F10 (0.33) SMN1; SMN2ALDH1A1HSD17B10OPRM1
SCHEMBL9735486 0.87 ALOX5 (0.36) ALOX5PDK2NPC1IDH1RAB9A
SCHEMBL8090273 0.87 RAB9A (0.34) ALOX5NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL7277059 0.85 KDM4E (0.35) ALOX5NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL8084985 0.84
SCHEMBL7269286 0.82 KMT2A (0.38) SMN1; SMN2ALDH1A1LMNAHSD17B10OPRM1
SCHEMBL8085187 0.81 LMNA (0.39) SMN1; SMN2LMNA
SCHEMBL8085204 0.81 KCNE1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed