SCHEMBL8090129

SCHEMBL8090129

COC12CCC(c3ccc(C(=O)N[CH]CCCNC(=N)N)cc3)(CC1)CC2

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
SPHK1 Q9NYA1 10/20 0.33
SPHK2 Q9NRA0 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
POLB P06746 2/20 0.32
HDAC3 O15379 1/20 0.31
F10 P00742 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091494 0.90 SPHK1 (0.34) ALDH1A1SPHK1SPHK2NPC1RAB9A
SCHEMBL8090161 0.87 SPHK1 (0.33) SPHK1SPHK2F10
SCHEMBL8090137 0.87 NPC1 (0.45) ALDH1A1NPC1RAB9APOLBHDAC3
SCHEMBL8091620 0.86 ALDH1A1 (0.32) ALDH1A1
SCHEMBL8083447 0.86 SPHK1 (0.33) SPHK1SPHK2F10
SCHEMBL8098109 0.86 ALDH1A1 (0.33) ALDH1A1NPC1RAB9APOLB
SCHEMBL8091469 0.86 ADRA1D (0.33) ALDH1A1RAB9A
SCHEMBL8098085 0.86 SPHK1 (0.33) ALDH1A1SPHK1SPHK2NPC1RAB9A
SCHEMBL8097998 0.85 SPHK1 (0.35) SPHK1SPHK2F10
SCHEMBL8091664 0.85 POLB (0.33) ALDH1A1SPHK1SPHK2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792883-B1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-12-20 EP claimed
EP-0792883-A1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-09-03 EP claimed
EP-0792883-B1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-12-20 EP disclosed
EP-0792883-A1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-09-03 EP disclosed