SCHEMBL8090541

SCHEMBL8090541

CC(=O)c1ccc2c(c1)C(n1nc(O)ccc1=O)C(C)(O)C(C)(C)O2

nearest known ligand 0.36

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085421 0.91 HTR1A (0.32)
SCHEMBL8084465 0.89 CA12 (0.35)
SCHEMBL8085200 0.88
SCHEMBL8088383 0.82 ALDH1A1 (0.36) AKR1B1
SCHEMBL8090511 0.82 ABCC9 (0.40)
SCHEMBL10697890 0.80 ABCC9 (0.41)
SCHEMBL8084238 0.77 AKR1B1 (0.30) AKR1B1
SCHEMBL8088411 0.76 KDM4E (0.33)
SCHEMBL8085312 0.71 ABCC9 (0.40)
SCHEMBL8090585 0.69 ABCC9 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed