SCHEMBL8084465

SCHEMBL8084465

COC(=O)c1ccc2c(c1)C(n1nc(O)ccc1=O)C(C)(O)C(C)(C)O2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.35
CA9 Q16790 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
XDH P47989 1/20 0.35
CA14 Q9ULX7 1/20 0.35
ALOX5 P09917 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
MAPT P10636 3/20 0.33
LMNA P02545 3/20 0.33
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8076906 0.89 ALDH1A1 (0.39) CA12CA9CA1CA2CA7
SCHEMBL8090541 0.89 AKR1B1 (0.32)
SCHEMBL8085421 0.88 HTR1A (0.32) TSHR
SCHEMBL8085200 0.85
SCHEMBL10696820 0.81 ABCC9 (0.39) LMNA
SCHEMBL8090511 0.80 ABCC9 (0.40) LMNAKDM4E
SCHEMBL8090273 0.79 RAB9A (0.34) CA12CA9CA1CA2CA7
SCHEMBL8085342 0.78 ALOX5 (0.39) CA12CA9ALOX5SMN1; SMN2LMNA
SCHEMBL7334077 0.76 ALOX5 (0.34) CA12CA9CA1CA2CA7
SCHEMBL7277059 0.73 KDM4E (0.35) CA12CA9ALOX5SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed