SCHEMBL8090657

SCHEMBL8090657

CCOC(=O)c1nccn1C1Cc2cc(CN(C)C=O)ccc2C1=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.33
GABRA5 P31644 2/20 0.33
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
GAA P10253 3/20 0.32
HPGD P15428 3/20 0.32
HSD17B10 Q99714 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
GLA P06280 2/20 0.30
NPC1 O15118 1/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
RAB9A P51151 1/20 0.30
HTR1D P28221 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7846559 0.88
SCHEMBL8090133 0.85 KDM4E (0.33) GABRA1GABRA5KDM4EALDH1A1GAA
SCHEMBL8091069 0.84 TBXAS1 (0.36) GABRA1GABRA5KDM4EALDH1A1GAA
SCHEMBL8880656 0.83 METAP1 (0.38) GABRA1GABRA5KDM4EALDH1A1GAA
SCHEMBL8880066 0.81 HRH1 (0.43) GABRA1GABRA5ALDH1A1MEN1MAPT
SCHEMBL8880563 0.81 GABRG2 (0.38) GABRA1GABRA5KDM4EALDH1A1GAA
SCHEMBL8881385 0.81 GABRG2 (0.41) GABRA1GABRA5KDM4EALDH1A1GAA
SCHEMBL8097517 0.81 KMT2A (0.43) GABRA1GABRA5ALDH1A1HPGDHSD17B10
SCHEMBL8881176 0.81 CYP19A1 (0.43) GABRA1GABRA5KDM4EALDH1A1HSD17B10
SCHEMBL8317441 0.79 GABRA1 (0.41) GABRA1GABRA5KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057454-A USEFUL FOR TREATING OR PREVENTING ALL ISCHAEMIAS (SUCH AS FOCAL OR GLOBAL ISCHAEMIA) RESULTING FROM CEREBROVASCULAR DISORDERS RHONE-POULENC RORER S.A. (FR) 2000-05-02 US disclosed
US-5902803-A 5H,10H-imidazo 1,2-a!indeno 1,2-e!pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE-POULENC RORER S.A. (FR) 1999-05-11 US disclosed