SCHEMBL8090721

SCHEMBL8090721

CCOC(=O)c1cn(C2Cc3c(C(=O)NCc4ccccc4)cccc3C2=O)c(C(=O)OCC)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
MAPK10 P53779 2/20 0.38
ESR1 P03372 1/20 0.38
MAPT P10636 1/20 0.38
ALDH1A1 P00352 4/20 0.37
HPGD P15428 4/20 0.37
MEN1 O00255 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPK1 P28482 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
TP53 P04637 2/20 0.36
CREBBP Q92793 1/20 0.36
HSD17B10 Q99714 2/20 0.36
GLA P06280 1/20 0.36
BRD4 O60885 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836007 0.85 CHRNB2 (0.41) KMT2AMAPK10ESR1MAPTALDH1A1
SCHEMBL8013343 0.80 GAA (0.38) MAPTALDH1A1KDM4ERAB9AGABRA2
SCHEMBL8100183 0.79 GAA (0.36) KMT2AMEN1MAPK1TP53GABRA2
SCHEMBL8098030 0.79 ADORA2A (0.40) KMT2AMAPK10ESR1MAPTALDH1A1
SCHEMBL8649980 0.78 GABRA2 (0.45) KMT2AMAPTALDH1A1HPGDMEN1
SCHEMBL8099222 0.78 GAA (0.38) MAPTALDH1A1HPGDKDM4EHSD17B10
SCHEMBL8098047 0.78 GAA (0.36) KMT2AALDH1A1MEN1KDM4EGABRA2
SCHEMBL7820269 0.78 P2RY12 (0.37) KMT2AMEN1
SCHEMBL8098246 0.77 GAA (0.38) MAPTALDH1A1HPGDKDM4ENPSR1
SCHEMBL8011792 0.77 GAA (0.36) MAPTALDH1A1HPGDKDM4EGABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057454-A USEFUL FOR TREATING OR PREVENTING ALL ISCHAEMIAS (SUCH AS FOCAL OR GLOBAL ISCHAEMIA) RESULTING FROM CEREBROVASCULAR DISORDERS RHONE-POULENC RORER S.A. (FR) 2000-05-02 US disclosed
US-5902803-A 5H,10H-imidazo 1,2-a!indeno 1,2-e!pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE-POULENC RORER S.A. (FR) 1999-05-11 US disclosed