SCHEMBL8098030

SCHEMBL8098030

CCOC(=O)c1c[nH]c(C2Cc3c(C(=O)NCc4ccccc4)cccc3C2=O)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.40
ADORA1 P30542 2/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
CREBBP Q92793 1/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.39
ESR1 P03372 1/20 0.39
MAPK10 P53779 1/20 0.39
HPGD P15428 3/20 0.38
HSD17B10 Q99714 2/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 2/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
ROCK2 O75116 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7844395 0.85 ADORA2A (0.40) ADORA2AADORA1KDM4EALDH1A1CREBBP
SCHEMBL8090721 0.79 KMT2A (0.38) KDM4EALDH1A1CREBBPKMT2AMAPT
SCHEMBL8098023 0.76 NSD2 (0.39) ALDH1A1CREBBPKMT2AMAPTESR1
SCHEMBL7844391 0.74 CREBBP (0.41) KDM4EALDH1A1CREBBPKMT2AMAPT
SCHEMBL7835910 0.72 ALDH1A1 (0.43) ALDH1A1KMT2AMAPTHPGDPOLB
SCHEMBL7847145 0.72 JAK3 (0.34) KDM4EALDH1A1KMT2AMAPTHPGD
SCHEMBL8556215 0.72 CHRNB2 (0.40) KDM4EALDH1A1CREBBPKMT2AMAPT
SCHEMBL7843220 0.70 CHRNB2 (0.53) KDM4EALDH1A1CREBBPKMT2AHPGD
SCHEMBL8090662 0.69
SCHEMBL7836007 0.68 CHRNB2 (0.41) ALDH1A1CREBBPKMT2AMAPTESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057454-A USEFUL FOR TREATING OR PREVENTING ALL ISCHAEMIAS (SUCH AS FOCAL OR GLOBAL ISCHAEMIA) RESULTING FROM CEREBROVASCULAR DISORDERS RHONE-POULENC RORER S.A. (FR) 2000-05-02 US disclosed
US-5902803-A 5H,10H-imidazo 1,2-a!indeno 1,2-e!pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE-POULENC RORER S.A. (FR) 1999-05-11 US disclosed