SCHEMBL8090771

SCHEMBL8090771

O=C1CC2(CCN(CC3CN(Cc4ccc5ccccc5c4)CC3c3ccccc3)CC2)c2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 14/20 0.45
KDM1A O60341 1/20 0.45
MAOB P27338 1/20 0.45
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
KMT2A Q03164 1/20 0.38
OPRL1 P41146 1/20 0.38
CCR3 P51677 1/20 0.37
UTS2R Q9UKP6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090716 0.84 ADRA1D (0.43) CCR5OPRL1UTS2R
SCHEMBL4414466 0.83 KMT2A (0.51) KDM1AMAOBHTR2AHTR2CHTR2B
SCHEMBL7838241 0.82 CCR5 (0.50) CCR5
SCHEMBL7836260 0.76 CCR5 (0.60) CCR5
SCHEMBL7837491 0.75 CCR5 (0.54) CCR5HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL7826160 0.75 CCR5 (0.65) CCR5
SCHEMBL8082670 0.72 CCR5 (0.51) CCR5
SCHEMBL1713596 0.72 SIGMAR1 (0.59) HTR2AHTR2CHTR2BSIGMAR1KMT2A
SCHEMBL8089197 0.71 CCR5 (0.56) CCR5
SCHEMBL7838025 0.69 CCR5 (0.57) CCR5HTR2AHTR2CHTR2BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166037-A Pyrrolidine and piperidine modulators of chemokine receptor activity MERCK & CO., INC. (US) 2000-12-26 US disclosed