SCHEMBL8091088

SCHEMBL8091088

COC(=O)C[C@@H](NC(=O)OC(C)(C)C)C1CC2CCC1N2S(=O)(=O)c1cc(F)cc(F)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
AKR1C3 P42330 1/20 0.33
HSD11B1 P28845 2/20 0.32
RORC P51449 5/20 0.32
SLC6A3 Q01959 4/20 0.31
SLC6A2 P23975 3/20 0.31
SLC6A4 P31645 2/20 0.31
APP P05067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13078574 0.89 ALDH1A1 (0.35) ALDH1A1AKR1C3HSD11B1RORCAPP
SCHEMBL3752853 0.77 ALDH1A1 (0.39) ALDH1A1AKR1C3HSD11B1RORC
SCHEMBL3741594 0.76 MMP13 (0.41) ALDH1A1AKR1C3HSD11B1RORC
SCHEMBL13078576 0.70 DPP4 (0.37)
SCHEMBL8097461 0.68 DPP4 (0.41) RORC
SCHEMBL19640870 0.67 AKR1C3 (0.53) AKR1C3HSD11B1APP
SCHEMBL8092352 0.65 MGLL (0.37)
SCHEMBL13078813 0.65 CTSK (0.34)
SCHEMBL8089162 0.64 STS (0.50)
SCHEMBL13078578 0.64 CACNA1B (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037719-A1 NOVEL COMPOUNDS AS DIPEPTIDYL PEPTIDASE IV (DPP IV) INHIBITORS LUPIN LIMITED (IN) 2009-03-26 WO disclosed