SCHEMBL8091369

SCHEMBL8091369

CCNS(=O)(=O)c1ccc(NS(C)(=O)=O)c(Oc2ccc(Cl)cc2Br)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
PTGS1 P23219 3/20 0.47
PTGS2 P35354 3/20 0.47
CYP2C9 P11712 1/20 0.43
TP53 P04637 1/20 0.43
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
EPAS1 Q99814 2/20 0.41
CCR2 P41597 1/20 0.41
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
CYP19A1 P11511 1/20 0.39
VCAM1 P19320 1/20 0.39
PKM P14618 1/20 0.38
WDR5 P61964 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091401 0.89 PTGS1 (0.60) ALDH1A1PTGS1PTGS2CYP2C9TP53
SCHEMBL8091867 0.85 ALDH1A1 (0.47) ALDH1A1PTGS1PTGS2CYP2C9KMT2A
SCHEMBL8104912 0.78 PTGS1 (0.57) ALDH1A1PTGS1PTGS2CYP2C9TP53
SCHEMBL8523996 0.78 CCR2 (0.60) ALDH1A1PTGS1PTGS2CYP2C9KMT2A
SCHEMBL8480176 0.76 PTGS1 (0.60) ALDH1A1PTGS1PTGS2CYP2C9TP53
SCHEMBL8092102 0.76 PTGS1 (0.60) ALDH1A1PTGS1PTGS2CYP2C9TP53
SCHEMBL8107816 0.76 PTGS1 (0.52) PTGS1PTGS2TP53KMT2AMAPT
SCHEMBL8091464 0.76 PTGS2 (0.62) ALDH1A1PTGS1PTGS2CYP2C9TP53
SCHEMBL8481953 0.75 PTGS1 (0.59) ALDH1A1PTGS1PTGS2CYP2C9TP53
SCHEMBL8107162 0.75 PTGS1 (0.61) ALDH1A1PTGS1PTGS2CYP2C9TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed