SCHEMBL8091392

SCHEMBL8091392

NCCCC(NC(=O)C1(C(=O)NCCc2cccnc2)CCCC1)OBOC(CCCN)NC(=O)C1(C(=O)NCCc2cccnc2)CCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.38
CYP3A4 P08684 1/20 0.37
HRH1 P35367 2/20 0.37
HDAC8 Q9BY41 2/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
EPHX1 P07099 1/20 0.36
EPHX2 P34913 1/20 0.36
HTT P42858 1/20 0.35
FES P07332 1/20 0.35
RET P07949 1/20 0.35
MARK3 P27448 1/20 0.35
TYK2 P29597 1/20 0.35
FLT4 P35916 1/20 0.35
SYK P43405 1/20 0.35
CLK2 P49760 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
PARP1 P09874 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091395 0.94 CYP2A6 (0.37) CYP2A6CYP3A4HRH1HDAC8HDAC2
SCHEMBL8098060 0.90 EPHX1 (0.36) HDAC8HDAC2HDAC6EPHX1EPHX2
SCHEMBL8095466 0.89 CYP2C19 (0.39) CYP3A4EPHX1MEN1NPC1RAB9A
SCHEMBL8095266 0.86 MMP1 (0.39) CYP3A4MEN1KMT2A
SCHEMBL8090127 0.85 KDM4E (0.36) NPC1RAB9ASMN1; SMN2
SCHEMBL8098087 0.84 MMP8 (0.44) EPHX2NPC1KMT2A
SCHEMBL8098074 0.84 EPHX1 (0.35) HDAC8HDAC2HDAC6EPHX1EPHX2
SCHEMBL8090157 0.82 MTNR1A (0.41) PARP1RAB9ALMNA
SCHEMBL8095467 0.82 CYP3A4 (0.38) CYP3A4EPHX1MEN1NPC1RAB9A
SCHEMBL8095182 0.81 MMP8 (0.40) EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792883-B1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-12-20 EP disclosed
EP-0792883-A1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-09-03 EP disclosed