SCHEMBL8091529

SCHEMBL8091529

CC(C)(C)OC(=O)CN(CCN(CC(=O)OC(C)(C)C)C(Cc1ccc(O)cc1)CN(CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
OPRM1 P35372 9/20 0.36
OPRK1 P41145 6/20 0.36
OPRD1 P41143 5/20 0.36
NR1D1 P20393 4/20 0.36
NR1H3 Q13133 1/20 0.34
ESR1 P03372 2/20 0.33
ESR2 Q92731 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5374479 0.94 CTSS (0.38) CTSSCTSKOPRM1OPRK1OPRD1
SCHEMBL8957471 0.89 CA1 (0.38) CTSSCTSKOPRM1OPRK1OPRD1
SCHEMBL8090950 0.89 NR1D1 (0.45) OPRM1OPRK1OPRD1NR1D1
SCHEMBL8957382 0.87 CTSS (0.39) CTSSCTSKOPRM1OPRK1OPRD1
SCHEMBL8668171 0.87 ACACB (0.37) NR1D1
SCHEMBL3748687 0.84 NR1D1 (0.36) CTSSCTSKNR1D1NR1H3
SCHEMBL8090953 0.83 ATM (0.39) CTSSCTSKOPRM1OPRK1OPRD1
SCHEMBL7511620 0.82 CTSS (0.40) CTSSCTSKNR1D1NR1H3ESR1
SCHEMBL8671108 0.82 ACACB (0.40) NR1D1
SCHEMBL92706 0.81 ACACB (0.38) NR1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6039931-A Derivatized DTPA complexes, pharmaceutical agents containing these compounds, their use, and processes for their production SCHERING AKTIENGESELLSCHAFT (DE) 2000-03-21 US disclosed
US-5853699-A Use of tetra azacycle complexes as x-ray diagnostic agents for the liver and gallbladder SCHERING AKTIENGESELLSCHAFT (DE) 1998-12-29 US disclosed
US-5798092-A METAL COMPLEXES; CONTRAST AGENTS FOR MEDICAL IMAGING SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-25 US disclosed
EP-0794800-A1 USE OF CHELATE COMPOUNDS AS DIAGNOSTIC AGENTS IN THE X-RAY EXAMINATION OF LIVER AND BILE DUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1997-09-17 EP disclosed
EP-0794799-A2 USE OF METAL COMPLEXES AS LIVER AND GALL BLADDER RADIODIAGNOSIS AGENTS IN COMPUTER TOMOGRAPHY SCHERING AKTIENGESELLSCHAFT (DE) 1997-09-17 EP disclosed
WO-1996016678-A1 USE OF CHELATE COMPOUNDS AS DIAGNOSTIC AGENTS IN THE X-RAY EXAMINATION OF LIVER AND BILE DUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1996-06-06 WO disclosed
WO-1996016677-A2 USE OF METAL COMPLEXES AS LIVER AND GALL BLADDER RADIODIAGNOSIS AGENTS IN COMPUTER TOMOGRAPHY SCHERING AKTIENGESELLSCHAFT (DE) 1996-06-06 WO disclosed
EP-0405704-B1 DTPA-complexes derivatives, pharmaceutical compositions containing them, their use and process for their preparation SCHERING AG (DE) 1994-12-14 EP disclosed