SCHEMBL8091827

SCHEMBL8091827

Cc1cc(C)c(Oc2cc(S(N)(=O)=O)ccc2NS(C)(=O)=O)c(S(N)(=O)=O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.38
CA2 P00918 6/20 0.38
CA9 Q16790 6/20 0.38
CA12 O43570 2/20 0.38
CYP19A1 P11511 5/20 0.38
KDM4E B2RXH2 3/20 0.38
MEN1 O00255 1/20 0.38
MLNR O43193 1/20 0.38
LMNA P02545 1/20 0.38
MMP1 P03956 1/20 0.38
MPO P05164 1/20 0.38
CYP1A2 P05177 1/20 0.38
GLA P06280 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
TBXA2R P21731 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099526 0.81 CYP19A1 (0.42) CA1CA2CA9CA12CYP19A1
SCHEMBL14280459 0.79 MRGPRX1 (0.54) CA1CA2CA9CA12CYP19A1
SCHEMBL4575282 0.73 SOS1 (0.55) CA1CA2CA9CA12CYP19A1
SCHEMBL4575511 0.73 PTGS1 (0.57) CA1CA2CA9CA12CYP19A1
SCHEMBL8101831 0.72 MAPK1 (0.46) CA1CA2CA9CA12CYP19A1
SCHEMBL8107162 0.71 PTGS1 (0.61) CA1CA2CA9CYP19A1LMNA
SCHEMBL8107798 0.71 PTGS2 (0.56) CA1CA2CA9CA12CYP19A1
SCHEMBL8091326 0.69 CYP19A1 (0.67) CA1CA2CA9CA12CYP19A1
SCHEMBL27357250 0.68 KDM4E (0.52) CA1CA2CA9CA12KDM4E
SCHEMBL8481948 0.68 ALDH1A1 (0.49) CA1CA2CA9CA12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed
EP-0848703-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II Nycomed Austria GmbH (AT) 1998-06-24 EP disclosed
WO-1997003953-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 1997-02-06 WO disclosed