SCHEMBL8092374

SCHEMBL8092374

Nc1cc(C2(S(=O)(=O)c3ccccc3)CC2)nc(-c2ccc(NC(=O)NC3COC3)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 7/20 0.39
MTOR P42345 5/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
PIK3CA P42336 7/20 0.39
PIK3CG P48736 2/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
ATR Q13535 2/20 0.36
PIK3R1 P27986 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084833 0.91 CA12 (0.43) MAPTHTTCA12CA1CA2
SCHEMBL8091191 0.91 PIK3CA (0.40) PIK3CDMTORPIK3CAPIK3CGATR
SCHEMBL8090316 0.90 KDR (0.37) PIK3CDMTORPIK3CAPIK3CGKDM4E
SCHEMBL8090948 0.89 CA12 (0.41) MTORPIK3CAKDM4EMAPTHTT
SCHEMBL8084016 0.89 CA12 (0.41) MTORPIK3CAKDM4EMAPTHTT
SCHEMBL8084603 0.86 PIK3CA (0.46) PIK3CDMTORHDAC3HDAC1HDAC2
SCHEMBL8090246 0.86 PIK3CA (0.42) PIK3CDMTORPIK3CAPIK3CGKDM4E
SCHEMBL8091293 0.85 MAPT (0.42) MTORPIK3CAPIK3CGKDM4EMAPT
SCHEMBL8099405 0.85 EPHX1 (0.42) MTORPIK3CAKDM4EMAPTHTT
SCHEMBL8098812 0.84 NPC1 (0.43) MAPTHTTCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed