SCHEMBL8090316

SCHEMBL8090316

Nc1cc(C2(S(=O)(=O)c3ccccc3)CC2)nc(-c2ccc(NC(=O)NC3CNNC3)cc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.37
KIT P10721 2/20 0.37
FLT3 P36888 2/20 0.37
MAPT P10636 3/20 0.36
KDM4E B2RXH2 2/20 0.36
HTT P42858 1/20 0.36
ATR Q13535 1/20 0.36
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CNR2 P34972 1/20 0.34
PIK3CD O00329 4/20 0.34
IGF1R P08069 1/20 0.34
PIK3CA P42336 3/20 0.34
MTOR P42345 1/20 0.33
PIK3CG P48736 1/20 0.33
NAMPT P43490 1/20 0.33
TTK P33981 1/20 0.33
PIK3R1 P27986 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092374 0.90 PIK3CD (0.39) MAPTKDM4EHTTATRCA12
SCHEMBL8084833 0.90 CA12 (0.43) KDRKITFLT3MAPTHTT
SCHEMBL8090948 0.89 CA12 (0.41) KDRKITFLT3MAPTKDM4E
SCHEMBL8084016 0.89 CA12 (0.41) KDRKITFLT3MAPTKDM4E
SCHEMBL8091191 0.86 PIK3CA (0.40) ATRCA12CA1CA2CA9
SCHEMBL8090246 0.85 PIK3CA (0.42) MAPTKDM4EHTTCNR2PIK3CD
SCHEMBL8091293 0.84 MAPT (0.42) MAPTKDM4EHTTATRCA1
SCHEMBL8099405 0.84 EPHX1 (0.42) KDRKITFLT3MAPTKDM4E
SCHEMBL8098812 0.83 NPC1 (0.43) MAPTHTTCA12CA1CA2
SCHEMBL8106295 0.83 CA12 (0.42) MAPTKDM4EHTTCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed