SCHEMBL8090246

SCHEMBL8090246

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccccc4)CC3)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.42
MTOR P42345 4/20 0.42
PIK3CG P48736 4/20 0.42
MAPT P10636 4/20 0.42
KDM4E B2RXH2 3/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CYP2C19 P33261 1/20 0.38
AKT1 P31749 2/20 0.38
AKT2 P31751 2/20 0.38
BDKRB1 P46663 1/20 0.38
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
PIP4K2A P48426 1/20 0.38
PIP4K2B P78356 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096342 0.96 PIK3CA (0.41) PIK3CAMTORPIK3CGMAPTKDM4E
SCHEMBL8092637 0.92 KMT2A (0.42) PIK3CAMTORPIK3CGKMT2ACYP2C19
SCHEMBL8099749 0.91 MTOR (0.40) PIK3CAMTORPIK3CGKMT2ACDK1
SCHEMBL8097257 0.91 ALDH1A1 (0.41) PIK3CAMTORPIK3CGKMT2AMEN1
SCHEMBL8083973 0.90 ALDH1A1 (0.43) PIK3CAMTORPIK3CGKMT2AMEN1
SCHEMBL8106295 0.90 CA12 (0.42) PIK3CAMTORMAPTKDM4EHTT
SCHEMBL8099045 0.89 MAPT (0.39) PIK3CAMTORPIK3CGMAPTKDM4E
SCHEMBL8091293 0.89 MAPT (0.42) PIK3CAMTORPIK3CGMAPTKDM4E
SCHEMBL8089917 0.89 PIK3CA (0.39) PIK3CAMTORPIK3CGKMT2AALDH1A1
SCHEMBL8092385 0.88 PIK3CD (0.41) PIK3CAMTORPIK3CGMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed