SCHEMBL8092850

SCHEMBL8092850

CC(C)NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccncc4)CC3)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
ROCK2 O75116 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP3A5 P20815 1/20 0.41
NAMPT P43490 6/20 0.39
PIK3CA P42336 3/20 0.35
MTOR P42345 1/20 0.35
PIK3CG P48736 1/20 0.35
PIK3CD O00329 4/20 0.35
AAK1 Q2M2I8 1/20 0.34
GHSR Q92847 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106295 0.92 CA12 (0.42) CA12CA1CA2CA9ROCK2
SCHEMBL8099749 0.90 MTOR (0.40) NAMPTPIK3CAMTORPIK3CGPIK3CD
SCHEMBL8099812 0.89 NAMPT (0.44) ROCK2NAMPTPIK3CAPIK3CDAAK1
SCHEMBL8104053 0.88 CA2 (0.41) CA12CA1CA2CA9ROCK2
SCHEMBL8098188 0.87 CA12 (0.44) CA12CA1CA2CA9ROCK2
SCHEMBL8090868 0.87 MTOR (0.38) NAMPTPIK3CAMTORPIK3CGPIK3CD
SCHEMBL8089531 0.86 CA12 (0.43) CA12CA1CA2CA9ROCK2
SCHEMBL8083655 0.86 NAMPT (0.43) NAMPTPIK3CAPIK3CD
SCHEMBL8099405 0.85 EPHX1 (0.42) CA12CA1CA2CA9NAMPT
SCHEMBL8092294 0.85 ROCK2 (0.39) CA12CA1CA2CA9ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed