SCHEMBL8104053

SCHEMBL8104053

CC(C)NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4cc(F)cc(F)c4)CC3)n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
PIK3CA P42336 3/20 0.36
MTOR P42345 2/20 0.36
EIF2S1 P05198 1/20 0.35
EIF2AK3 Q9NZJ5 1/20 0.35
ROCK2 O75116 2/20 0.35
PIK3CD O00329 4/20 0.34
NAMPT P43490 2/20 0.34
GHSR Q92847 2/20 0.34
ABL1 P00519 1/20 0.34
MMP2 P08253 1/20 0.33
PIK3CG P48736 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP3A5 P20815 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LIMK1 P53667 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089917 0.90 PIK3CA (0.39) CA2CA9PIK3CAMTORPIK3CD
SCHEMBL8106295 0.89 CA12 (0.42) CA2CA9CA12CA1PIK3CA
SCHEMBL8104051 0.89 NAMPT (0.38) PIK3CAMTORPIK3CDNAMPT
SCHEMBL8092850 0.88 CA12 (0.42) CA2CA9CA12CA1PIK3CA
SCHEMBL8097966 0.87 KIF11 (0.37) PIK3CAMTORPIK3CDNAMPTPIK3CG
SCHEMBL8099487 0.86 CA12 (0.42) CA2CA9CA12CA1CYP3A4
SCHEMBL8089000 0.86 PIK3CD (0.40) CA2CA9CA12CA1PIK3CA
SCHEMBL8098188 0.86 CA12 (0.44) CA2CA9CA12CA1PIK3CA
SCHEMBL8089531 0.85 CA12 (0.43) CA2CA9CA12CA1PIK3CA
SCHEMBL8082005 0.85 PIK3CA (0.41) CA2CA9CA12CA1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed