SCHEMBL8093418

SCHEMBL8093418

COc1ccc(C(C(N)=O)(C(C)C)N2C(=O)C(N)C(C)(C)Sc3ccccc32)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.35
BCHE P06276 3/20 0.34
ACHE P22303 1/20 0.34
GSK3B P49841 2/20 0.34
LMNA P02545 4/20 0.33
KIF11 P52732 3/20 0.33
CYP3A4 P08684 3/20 0.33
TSHR P16473 2/20 0.33
ABCB11 O95342 2/20 0.33
KCNH2 Q12809 2/20 0.33
SLC22A1 O15245 1/20 0.33
CACNA1F O60840 1/20 0.33
ABCB1 P08183 1/20 0.33
HRH2 P25021 1/20 0.33
ADRA1A P35348 1/20 0.33
SCN1A P35498 1/20 0.33
SCN4A P35499 1/20 0.33
HTT P42858 1/20 0.33
SCN7A Q01118 1/20 0.33
CACNA1D Q01668 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8405727 0.77 BRD4 (0.38) MAPTALDH1A1MEN1KMT2AHDAC2
SCHEMBL8405648 0.73 ALDH1A1 (0.33) MAPTLMNAKIF11TSHRALDH1A1
SCHEMBL8519231 0.72 GAA (0.37) MAPTLMNAALDH1A1HPGD
SCHEMBL8406820 0.72 KMT2A (0.39) MAPTLMNACYP3A4ALDH1A1MEN1
SCHEMBL8816172 0.71 KIF11 (0.35) MAPTLMNAKIF11ALDH1A1MEN1
SCHEMBL8812237 0.70 CCKAR (0.40) MAPTKIF11ALDH1A1KMT2A
SCHEMBL8406772 0.69 POLB (0.33) ALDH1A1
SCHEMBL8814705 0.67 CCKAR (0.49) MAPTALDH1A1MEN1KMT2A
SCHEMBL8813766 0.66 CCKAR (0.39)
SCHEMBL8797930 0.66 HDAC3 (0.51) SCN9AHDAC3HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096885-A EXHIBIT AGONIST ACTIVITY FOR CCK-A RECEPTORS THEREBY ENABLING THEM TO MODULATE THE HORMONES GASTRIN AND CHOLECYSTOKININ IN MAMMALS. GLAXO WELLCOME INC. (US) 2000-08-01 US disclosed