SCHEMBL8405648

SCHEMBL8405648

COc1ccc(C(C(N)=O)(C(C)C)N2C(=O)C(N)C(=O)N(c3ncccn3)c3ccccc32)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 2/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
F2 P00734 1/20 0.32
CCKAR P32238 1/20 0.32
CCKBR P32239 1/20 0.32
NPC1 O15118 5/20 0.31
RAB9A P51151 5/20 0.31
CDK5 Q00535 2/20 0.31
PAX8 Q06710 2/20 0.31
CDK5R1 Q15078 2/20 0.31
PKM P14618 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
AHR P35869 1/20 0.31
HPGD P15428 1/20 0.31
SLC6A7 Q99884 1/20 0.31
MC4R P32245 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8406820 0.91 KMT2A (0.39) ALDH1A1KDM4EKMT2AALOX15HSD17B10
SCHEMBL8519231 0.86 GAA (0.37) ALDH1A1CCKARCCKBRRAB9AHPGD
SCHEMBL8406772 0.83 POLB (0.33) ALDH1A1CCKARCCKBR
SCHEMBL8405727 0.78 BRD4 (0.38) ALDH1A1KDM4EKMT2AHSD17B10CCKBR
SCHEMBL7753002 0.78 CCKBR (0.37) ALDH1A1KMT2ACCKARCCKBRRAB9A
SCHEMBL8816172 0.74 KIF11 (0.35) ALDH1A1KMT2ACCKARCCKBRHPGD
SCHEMBL8093418 0.73 MAPT (0.35) ALDH1A1KMT2AHPGDLMNATSHR
SCHEMBL8814705 0.71 CCKAR (0.49) ALDH1A1KMT2ACCKARCCKBRPKM
SCHEMBL8402034 0.71 CCKAR (0.57) CCKARCCKBR
SCHEMBL8813766 0.71 CCKAR (0.39) CCKARCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0756602-B1 CCK OR GASTRIN MODULATING 5-HETEROCYCLIC-1,5-BENZODIAZEPINES GLAXO WELLCOME INC (US) 1999-06-30 EP disclosed