SCHEMBL8092670

SCHEMBL8092670

CCOC(=O)CNc1nc(-c2ccc(F)cc2)c(-c2ccc(S(N)(=O)=O)cc2)cc1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.44
CHRNA7 P36544 6/20 0.44
PTGS2 P35354 4/20 0.43
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 5/20 0.42
L3MBTL1 Q9Y468 5/20 0.42
HPGD P15428 4/20 0.42
LMNA P02545 4/20 0.42
TDP1 Q9NUW8 3/20 0.42
NPSR1 Q6W5P4 3/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA4 P22748 1/20 0.42
GAA P10253 1/20 0.41
ALOX15 P16050 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8094729 0.92 PTGS2 (0.49) GLAPTGS2KDM4EALDH1A1L3MBTL1
SCHEMBL8776744 0.86 SQOR (0.46) GLACHRNA7PTGS2KDM4EL3MBTL1
SCHEMBL8095872 0.83 ALDH1A1 (0.55) PTGS2KDM4EALDH1A1L3MBTL1HPGD
SCHEMBL8093864 0.83 CA9 (0.44) CHRNA7PTGS2CA1CA2CA9
SCHEMBL8086911 0.82 HPGD (0.45) PTGS2KDM4EALDH1A1L3MBTL1HPGD
SCHEMBL8094551 0.80 CNR1 (0.49) PTGS2L3MBTL1NPSR1CA1CA2
SCHEMBL8093983 0.80 CNR1 (0.44) CHRNA7PTGS2KDM4EL3MBTL1CA1
SCHEMBL8421064 0.79 ALDH1A1 (0.49) GLAKDM4EALDH1A1L3MBTL1HPGD
SCHEMBL8093987 0.79 PTGS2 (0.48) PTGS2CA1CA2CA9PTGS1
SCHEMBL8094187 0.78 CNR1 (0.50) PTGS2CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed