SCHEMBL8094532

SCHEMBL8094532

CC(C)(C)c1cc(C2CNC(=O)N2C(=O)c2ccc(N)cc2)cc(C(C)(C)C)c1O

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 2/20 0.36
ALPL P05186 2/20 0.36
XIAP P98170 2/20 0.36
NR1H4 Q96RI1 1/20 0.36
ALOX5 P09917 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
F2R P25116 1/20 0.34
HSP90AA1 P07900 4/20 0.33
HSP90AB1 P08238 4/20 0.33
MAOB P27338 2/20 0.33
GAA P10253 1/20 0.32
NISCH Q9Y2I1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104050 0.85 SMN1; SMN2 (0.44) NR1H4
SCHEMBL8094518 0.79 ALOX5 (0.43) ALOX5PTGS1PTGS2GAA
SCHEMBL4325286 0.68 NR1H4 (0.38) ENPP3ALPLXIAPNR1H4ALOX5
SCHEMBL10449344 0.67 ALOX5 (0.55) NR1H4ALOX5PTGS1PTGS2F2R
SCHEMBL4315862 0.64 F2R (0.32) NR1H4F2RMAOBGAA
SCHEMBL4319085 0.63 ALDH1A1 (0.47)
SCHEMBL4319308 0.63 ALDH1A1 (0.54) HSP90AA1HSP90AB1GAA
SCHEMBL4319185 0.60 SNCA (0.65) NR1H4PTGS1GAA
SCHEMBL9524225 0.60 CA2 (0.68) PTGS1PTGS2NISCH
SCHEMBL7018969 0.60 CYP19A1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991654-A1 NOVEL 2-(IMINOMETHYL)AMINO-PHENYL DERIVATIVES, PREPARATION, APPLICATION AS MEDICINES AND COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2000-04-12 EP disclosed
WO-1998058934-A1 NOVEL 2-(IMINOMETHYL)AMINO-PHENYL DERIVATIVES, PREPARATION, APPLICATION AS MEDICINES AND COMPOSITIONS CONTAINING SAME SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1998-12-30 WO disclosed