SCHEMBL8094653

SCHEMBL8094653

Cc1cc(CC2CCN(Cc3ccc(F)c(C#N)c3)CC2)c2ccccc2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.47
HTR2B P41595 1/20 0.45
NCF1 P14598 1/20 0.43
CHRM4 P08173 4/20 0.43
CHRM2 P08172 3/20 0.43
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
JAK3 P52333 1/20 0.42
ATM Q13315 2/20 0.42
CHRM1 P11229 2/20 0.41
ACHE P22303 2/20 0.41
ALDH1A1 P00352 2/20 0.41
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13945424 0.84 HTR1D (0.47) PDE2AHTR2BNCF1CHRM4JAK2
SCHEMBL8091569 0.79 CYP3A4 (0.49) CHRM4ATMALDH1A1
SCHEMBL8092993 0.77 HTR2B (0.44) HTR2BCHRM4ATMACHE
SCHEMBL8096499 0.77 GAA (0.53) NCF1ACHEGAABCHE
SCHEMBL8095852 0.73 CCR3 (0.47) ATMALDH1A1KDM4EMAPTHTT
SCHEMBL27822767 0.72 DPP4 (0.57) PDE2AHTR2BCHRM4CHRM2JAK2
SCHEMBL8103772 0.70 DPP4 (0.43) ATMCHRM1ACHEALDH1A1KDM4E
SCHEMBL1935654 0.70 ALDH1A1 (0.63) PDE2AHTR2BNCF1JAK2JAK1
SCHEMBL29668952 0.70 CHKA (0.62) PDE2AHTR2BJAK2JAK1JAK3
SCHEMBL20238481 0.70 CHKA (0.62) PDE2AHTR2BJAK2JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000085-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES USEFUL AS MODULATORS OF GATED ION CHANNELS PAINCEPTOR PHARMA CORPORATION (CA) 2008-12-31 WO disclosed