SCHEMBL8094729

SCHEMBL8094729

CCOC(=O)CNc1nc(-c2ccc(F)cc2)c(-c2ccc(S(C)(=O)=O)cc2)cc1C#N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.49
PTGS1 P23219 1/20 0.47
GLA P06280 1/20 0.45
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 4/20 0.43
L3MBTL1 Q9Y468 4/20 0.43
LMNA P02545 3/20 0.43
TDP1 Q9NUW8 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
GAA P10253 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092670 0.92 GLA (0.44) PTGS2PTGS1GLAKDM4EALDH1A1
SCHEMBL8099443 0.84 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL8086508 0.84 PTGS2 (0.60) PTGS2PTGS1KDM4EALDH1A1HPGD
SCHEMBL8095119 0.82 HPGD (0.47) PTGS2PTGS1KDM4EALDH1A1HPGD
SCHEMBL8094067 0.81 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL8421064 0.80 ALDH1A1 (0.49) GLAKDM4EALDH1A1HPGDL3MBTL1
SCHEMBL8100740 0.80 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL8095481 0.80 PTGS2 (0.54) PTGS2PTGS1KDM4EL3MBTL1
SCHEMBL8099266 0.80 PTGS2 (0.53) PTGS2PTGS1ALDH1A1
SCHEMBL8101771 0.79 PTGS2 (0.54) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed