SCHEMBL8094989

SCHEMBL8094989

CCCCOC(=O)COc1nc(-c2ccc(F)cc2)c(-c2ccc(S(N)(=O)=O)cc2)cc1C#N

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.53
PTGS1 P23219 1/20 0.53
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CNR1 P21554 8/20 0.41
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 3/20 0.39
TSHR P16473 1/20 0.39
CA7 P43166 1/20 0.39
CHRNA7 P36544 3/20 0.38
CNR2 P34972 1/20 0.38
SQOR Q9Y6N5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8086366 0.92 PTGS2 (0.63) PTGS2PTGS1MEN1KMT2ANPSR1
SCHEMBL8776744 0.91 SQOR (0.46) PTGS2PTGS1MEN1KMT2ANPSR1
SCHEMBL8094547 0.91 PTGS2 (0.60) PTGS2PTGS1MEN1KMT2ANPSR1
SCHEMBL8095632 0.89 PTGS2 (0.56) PTGS2PTGS1CNR1CA12CA1
SCHEMBL8092530 0.88 PTGS2 (0.55) PTGS2PTGS1MEN1KMT2ANPSR1
SCHEMBL8093983 0.88 CNR1 (0.44) PTGS2PTGS1L3MBTL1CNR1CA12
SCHEMBL8094551 0.85 CNR1 (0.49) PTGS2PTGS1MEN1KMT2ANPSR1
SCHEMBL8087099 0.83 PTGS2 (0.48) PTGS2PTGS1MEN1KMT2ACNR1
SCHEMBL8093419 0.83 PTGS2 (0.72) PTGS2PTGS1CNR1CNR2
SCHEMBL8095681 0.82 CA2 (0.51) PTGS2PTGS1CNR1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed